Products >> Drug Discovery >> Assay/Kits >> Assays (CIS BIO) >> GPCR
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GPCR

Kinases

Biomarkers

Assays on Demand

Custom Labelling

GPCR Solutions

Comprehensive HTRF cellular platform

Cell surface receptor studies and functional assays.

GPCR investigation is among the top priorities in drug discovery research.

Cisbio has supported this area for many years by bringing regularly cutting edge assays and technologies fitted for receptor characterization and for compounds screening and lead optimization

Cisbio expands its offers for functional readouts (second messenger accumulation assays: cyclic-AMP & IP-One) with Cellul'erk, a new assay which allows detection of phosphorylated ERK directly in cells.

The new Tag-lite™ cell-surface receptor platform means Cisbio Bioassays now provides reagents and technology to address the latest evolution in the GPCR drug discovery field.

 

 

Applications:
 

Binding assays

GPCR dimer assays
GPCR functional assays:
  - Second messenger assays (cAMP & IP-One)
- The first HTRF Phospho-ER1/2 assay
 

Features:

Single technology and cellular platform for all GPCR assays

Unique non-radioactive ligand binding assays
Miniaturization down to < 10µl

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